Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04110
Ion Channel
Glutamate receptor ionotropic subunit NMDA 1
Peptide Function
Inhibitor
Gene Name
Grin1
Activity Data (nM)
IC50
487 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GEγγLQγNQγLIRγKSN-NH2
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
[Conotoxin GV; Conotoxin G V; 93438-65-4; Sleeper peptide; Snail sleeper peptide; Conantokin-G; Conantokin G; UNII-32CFR9L3TD; CGX-1007; 32CFR9L3TD; Conotoxin G V;GEXXLQXNQX LIRXKSN; DTXSID10896916; AKOS024457994; NS00075388]
Peptide Species
Conus geographus (Geography cone) (Nubecula geographus)
Peptide Name
Conantokin-G (con-G)
CAS Number
93438-65-4
Experimental Conditions
pH
pH 7.35
Holding Potential (mV)
−70 mV
Temperature
Room Temperture
Test Method
Patch-clamping
Test Species
Murine hippocampal 16-day embryonic neurons
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
i-GluRs
Ion Channel UniProt Accession
Source Organism
Mus musculus (Mouse)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available